Solid-phase synthesis of 1,2,3, 4-tetrahydro-beta-carboline-containing peptidomimetics.

نویسندگان

  • X Li
  • L Zhang
  • W Zhang
  • S E Hall
  • J P Tam
چکیده

A solid-phase method for the synthesis of 1,2,3, 4-tetrahydro-beta-carboline-containing peptidomimetics has been developed. The key step in the strategy is the Pictet-Spengler condensation of a resin-bound tryptophan-containing fragment with an Fmoc-amino aldehyde.

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عنوان ژورنال:
  • Organic letters

دوره 2 20  شماره 

صفحات  -

تاریخ انتشار 2000